|
[11] Number: | 1 -2003-500145 | Document Code: PH B1 |
[45] Issued: | 6/28/2007 |
[54] Title: | NOVEL NON-IMIDAZOLE COMPOUNDS |
[72] Inventor(s): |
NENG-YANG SHIH, OF NEW JERSEY, UNITED STATES OF AMERICA CHRISTOPHER W BOYCE, OF NEW JERSEY, UNITED STATES OF AMERICA MWANGI WA MUTAHI, OF NEW JERSEY, UNITED STATES OF AMERICA JOHN J PIWINSKI, OF NEW JERSEY, UNITED STATES OF AMERICA ROBERT G ASLANIAN, OF NEW JERSEY, UNITED STATES OF AMERICA MICHAEL Y BERLIN, OF NEW JERSEY, UNITED STATES OF AMERICA PIETRO MANGIARACINA, OF NEW YORK, UNITED STATES OF AMERICA PAULINE C TING, OF NEW JERSEY, UNITED STATES OF AMERICA STUART B ROSENBLUM, OF NEW JERSEY, UNITED STATES OF AMERICA KEVIN D McCORMICK, OF NEW JERSEY, UNITED STATES OF AMERICA WING C TOM, OF NEW JERSEY, UNITED STATES OF AMERICA |
[73] Applicant/Assignee(s): |
SCHERING CORPORATION , OF NEW JERSEY, UNITED STATES OF AMERICA |
[74] Attorney/Agent: | SIGUION REYNA ET AL |
[22] Date Filed: | 3/19/2003 |
[21] Application Serial Number: | 1- 2003-500145 |
[30] | Priority Data: | ||||||||
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Disclosed are novel compounds of the formula: (I) Also
disclosed are pharmaceutical compositions comprising the compounds of
Formula (I). Also disclosed are methods of treating various diseases or
conditions, such as, for example, allergy, allergy-induced airway responses,
and congestion (e.g., nasal congestion) using the compounds of Formula (I).
Also disclosed are methods of treating various diseases or conditions, such
as, for example, allergy, allergy-induced airway responses, and congestion
(e,g., nasal congestion) using the compounds of Formula (I) in combination
with a H1 receptor antagonist.
[52] PH
Class: NONE
[51]
International Class7:
A61K 31/4545; A61K 31/506; A61P 3/04; C07D 213/73; C07D 401/12; C07D 409/14; C07D 413/14; C07D 417/14; C07D 498/04; A61K 31/4985; A61K 31/4523; C07D 401/14; A61P 37/08
[58] Field
of Search:
A61K 31/4545; A61K 31/506; A61P 3/04; C07D 213/73; C07D 401/12; C07D 409/14; C07D 413/14; C07D 417/14; C07D 498/04; A61K 31/4985; A61K 31/4523; C07D 401/14; A61P 37/08
[56] Reference(s)
Cited and/or Considered: NONE
[57] Abstract:
No.
of Claims: 246